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<front>
<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Front cover</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/C1MD90010B</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Author</surname><given-names>Anonymous</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>219</fpage>
<lpage>219</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=C1MD90010B">Abstract</self-uri>
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<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Inside front cover</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/C1MD90011K</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Author</surname><given-names>Anonymous</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>220</fpage>
<lpage>220</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=C1MD90011K">Abstract</self-uri>
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<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Contents</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/C1MD90012A</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Author</surname><given-names>Anonymous</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>221</fpage>
<lpage>228</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=C1MD90012A">Abstract</self-uri>
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<article>
<front>
<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Natural products targeting telomere maintenance</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00241k</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Chen</surname>
<given-names>Jack Li-Yang</given-names></name>
<name><surname>Sperry</surname>
<given-names>Jonathan</given-names></name>
<name><surname>Ip</surname>
<given-names>Nancy Y.</given-names></name>
<name><surname>Brimble</surname>
<given-names>Margaret A.</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>229</fpage>
<lpage>245</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00241k">Abstract</self-uri>
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</article>
<article>
<front>
<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>The p53-MDM2/MDMX axis – A chemotype perspective</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00248h</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Khoury</surname>
<given-names>Kareem</given-names></name>
<name><surname>Popowicz</surname>
<given-names>Grzegorz M.</given-names></name>
<name><surname>Holak</surname>
<given-names>Tad A.</given-names></name>
<name><surname>Dömling</surname>
<given-names>Alexander</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>246</fpage>
<lpage>260</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00248h">Abstract</self-uri>
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</article>
<article>
<front>
<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Conformational effects on potency of thioimidazoles and dihydrothiazolines</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00228c</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Selig</surname>
<given-names>Roland</given-names></name>
<name><surname>Schattel</surname>
<given-names>Verena</given-names></name>
<name><surname>Goettert</surname>
<given-names>Marcia</given-names></name>
<name><surname>Schollmeyer</surname>
<given-names>Dieter</given-names></name>
<name><surname>Albrecht</surname>
<given-names>Wolfgang</given-names></name>
<name><surname>Laufer</surname>
<given-names>Stefan</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>261</fpage>
<lpage>269</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00228c">Abstract</self-uri>
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</article>
<article>
<front>
<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Preparation of blood-brain barrier-permeable paclitaxel-carrier conjugate and its chemotherapeutic activity in the mouse glioblastoma model</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00235f</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Jin</surname>
<given-names>Juyoun</given-names></name>
<name><surname>Lee</surname>
<given-names>Woo Sirl</given-names></name>
<name><surname>Joo</surname>
<given-names>Kyeung Min</given-names></name>
<name><surname>Maiti</surname>
<given-names>Kaustabh K.</given-names></name>
<name><surname>Biswas</surname>
<given-names>Goutam</given-names></name>
<name><surname>Kim</surname>
<given-names>Wanil</given-names></name>
<name><surname>Kim</surname>
<given-names>Kyong-Tai</given-names></name>
<name><surname>Lee</surname>
<given-names>Se Jeong</given-names></name>
<name><surname>Kim</surname>
<given-names>Kang-Ho</given-names></name>
<name><surname>Nam</surname>
<given-names>Do-Hyun</given-names></name>
<name><surname>Chung</surname>
<given-names>Sung-Kee</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>270</fpage>
<lpage>273</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00235f">Abstract</self-uri>
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</article>
<article>
<front>
<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Platinum-oxazoline complexes as anti-cancer agents: syntheses, characterisation and initial biological studies</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00211a</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Yadav</surname>
<given-names>Paras N.</given-names></name>
<name><surname>Beveridge</surname>
<given-names>Ramsay E.</given-names></name>
<name><surname>Blay</surname>
<given-names>Jonathan</given-names></name>
<name><surname>Boyd</surname>
<given-names>Alaina R.</given-names></name>
<name><surname>Chojnacka</surname>
<given-names>Maja W.</given-names></name>
<name><surname>Decken</surname>
<given-names>Andreas</given-names></name>
<name><surname>Deshpande</surname>
<given-names>Ankur A.</given-names></name>
<name><surname>Gardiner</surname>
<given-names>Michael G.</given-names></name>
<name><surname>Hambley</surname>
<given-names>Trevor W.</given-names></name>
<name><surname>Hughes</surname>
<given-names>Michael J.</given-names></name>
<name><surname>Jolly</surname>
<given-names>Leslie</given-names></name>
<name><surname>Lavangie</surname>
<given-names>Jacquelyn A.</given-names></name>
<name><surname>MacInnis</surname>
<given-names>Timothy D.</given-names></name>
<name><surname>McFarland</surname>
<given-names>Sherri A.</given-names></name>
<name><surname>New</surname>
<given-names>Elizabeth J.</given-names></name>
<name><surname>Gossage</surname>
<given-names>Robert A.</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>274</fpage>
<lpage>277</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00211a">Abstract</self-uri>
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</article>
<article>
<front>
<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>New insight into the mode of action of vancomycin dimers in bacterial cell wall synthesis</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00230e</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Yoshida</surname>
<given-names>Osamu</given-names></name>
<name><surname>Nakamura</surname>
<given-names>Jun</given-names></name>
<name><surname>Yamashiro</surname>
<given-names>Hidenori</given-names></name>
<name><surname>Miura</surname>
<given-names>Kenji</given-names></name>
<name><surname>Hayashi</surname>
<given-names>Sayaka</given-names></name>
<name><surname>Umetsu</surname>
<given-names>Kosei</given-names></name>
<name><surname>Xu</surname>
<given-names>Shu</given-names></name>
<name><surname>Maki</surname>
<given-names>Hideki</given-names></name>
<name><surname>Arimoto</surname>
<given-names>Hirokazu</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>278</fpage>
<lpage>282</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00230e">Abstract</self-uri>
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<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Interaction mechanisms of CdTe quantum dots with proteins possessing different isoelectric points</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00237b</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Lu</surname>
<given-names>Zhisong</given-names></name>
<name><surname>Hu</surname>
<given-names>Weihua</given-names></name>
<name><surname>Bao</surname>
<given-names>Haifeng</given-names></name>
<name><surname>Qiao</surname>
<given-names>Yan</given-names></name>
<name><surname>Li</surname>
<given-names>Chang Ming</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>283</fpage>
<lpage>286</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00237b">Abstract</self-uri>
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<front>
<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Oxazole phosphonic acids as fructose 1,6-bisphosphatase inhibitors with potent glucose-lowering activity</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00269k</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Dang</surname>
<given-names>Qun</given-names></name>
<name><surname>Kasibthatla</surname>
<given-names>Srinivas Rao</given-names></name>
<name><surname>Jiang</surname>
<given-names>Tao</given-names></name>
<name><surname>Taplin</surname>
<given-names>Frank</given-names></name>
<name><surname>Gibson</surname>
<given-names>Tony</given-names></name>
<name><surname>Potter</surname>
<given-names>Scott C.</given-names></name>
<name><surname>Poelje</surname>
<given-names>Paul D. van</given-names></name>
<name><surname>Erion</surname>
<given-names>Mark D.</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>287</fpage>
<lpage>290</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00269k">Abstract</self-uri>
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<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Potent sirtuin inhibition bestowed by l-2-amino-7-carboxamidoheptanoic acid (l-ACAH), a N&lt;sup&gt;ε&lt;/sup&gt;-acetyl-lysine analog</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00212g</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Hirsch</surname>
<given-names>Brett M.</given-names></name>
<name><surname>Du</surname>
<given-names>Zhanwen</given-names></name>
<name><surname>Li</surname>
<given-names>Xiaopeng</given-names></name>
<name><surname>Sylvester</surname>
<given-names>Jorge A.</given-names></name>
<name><surname>Wesdemiotis</surname>
<given-names>Chrys</given-names></name>
<name><surname>Wang</surname>
<given-names>Zhenghe</given-names></name>
<name><surname>Zheng</surname>
<given-names>Weiping</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>291</fpage>
<lpage>299</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00212g">Abstract</self-uri>
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<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Extended side chain analogues of 8-aminoquinolines: Synthesis and evaluation of antiprotozoal, antimicrobial, β-hematin inhibition, and cytotoxic activities</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00267d</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Kaur</surname>
<given-names>Kirandeep</given-names></name>
<name><surname>Jain</surname>
<given-names>Meenakshi</given-names></name>
<name><surname>Khan</surname>
<given-names>Shabana I.</given-names></name>
<name><surname>Jacob</surname>
<given-names>Melissa R.</given-names></name>
<name><surname>Tekwani</surname>
<given-names>Babu L.</given-names></name>
<name><surname>Singh</surname>
<given-names>Savita</given-names></name>
<name><surname>Singh</surname>
<given-names>Prati Pal</given-names></name>
<name><surname>Jain</surname>
<given-names>Rahul</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>300</fpage>
<lpage>307</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00267d">Abstract</self-uri>
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<front>
<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Structure and antimicrobial properties of multivalent short peptides</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00247j</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Young</surname>
<given-names>Anne W.</given-names></name>
<name><surname>Liu</surname>
<given-names>Zhigang</given-names></name>
<name><surname>Zhou</surname>
<given-names>Chunhui</given-names></name>
<name><surname>Totsingan</surname>
<given-names>Filbert</given-names></name>
<name><surname>Jiwrajka</surname>
<given-names>Nikhil</given-names></name>
<name><surname>Shi</surname>
<given-names>Zhengshuang</given-names></name>
<name><surname>Kallenbach</surname>
<given-names>Neville R.</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>308</fpage>
<lpage>314</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00247j">Abstract</self-uri>
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<article>
<front>
<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Diphenylbutylpiperidine-based cell autophagy inducers: Design, synthesis and SAR studies</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00236d</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Chen</surname>
<given-names>Gang</given-names></name>
<name><surname>Xia</surname>
<given-names>Hongguang</given-names></name>
<name><surname>Cai</surname>
<given-names>Yu</given-names></name>
<name><surname>Ma</surname>
<given-names>Dawei</given-names></name>
<name><surname>Yuan</surname>
<given-names>Junying</given-names></name>
<name><surname>Yuan</surname>
<given-names>Chengye</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>315</fpage>
<lpage>320</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00236d">Abstract</self-uri>
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</article>
<article>
<front>
<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Water soluble flavonol prodrugs that protect against ischaemia-reperfusion injury in rat hindlimb and sheep heart</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00240b</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Williams</surname>
<given-names>Spencer J.</given-names></name>
<name><surname>Thomas</surname>
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<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>321</fpage>
<lpage>324</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00240b">Abstract</self-uri>
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<front>
<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Development of a phosphatase-resistant, l-tyrosine derived LPA1/LPA3 dual antagonist</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00273a</article-id><contrib-group><contrib contrib-type="author">
<name><surname>East</surname>
<given-names>James E.</given-names></name>
<name><surname>Carter</surname>
<given-names>Karen M.</given-names></name>
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<given-names>Perry C.</given-names></name>
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<given-names>Nancy A.</given-names></name>
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<given-names>Myron L.</given-names></name>
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<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>325</fpage>
<lpage>330</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00273a">Abstract</self-uri>
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<front>
<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Erythromycin B: conformational analysis and antibacterial activity</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/c0md00251h</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Tyson</surname>
<given-names>Paul</given-names></name>
<name><surname>Hassanzadeh</surname>
<given-names>Abdolreza</given-names></name>
<name><surname>Mordi</surname>
<given-names>Mohd. Nizam</given-names></name>
<name><surname>Allison</surname>
<given-names>David G.</given-names></name>
<name><surname>Marquez</surname>
<given-names>Viter</given-names></name>
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</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>331</fpage>
<lpage>336</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=c0md00251h">Abstract</self-uri>
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<journal-meta>
<journal-title>MedChemComm</journal-title>
<issn>2040-2503</issn>
<publisher>
<publisher-name>Royal Society of Chemistry</publisher-name>
</publisher>
</journal-meta>
<article-meta>
<title-group>
<article-title>Back cover</article-title>
</title-group>
<article-id pub-id-type="doi">10.1039/C1MD90013G</article-id><contrib-group><contrib contrib-type="author">
<name><surname>Author</surname><given-names>Anonymous</given-names></name>
</contrib></contrib-group>
<pub-date pub-type="pub"><year>2011</year></pub-date>
<volume>2</volume>
<issue>4</issue>
<fpage>337</fpage>
<lpage>338</lpage>
<self-uri xlink:href="http://xlink.rsc.org/?DOI=C1MD90013G">Abstract</self-uri>
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