MedChemComm 2040-2503 Royal Society of Chemistry Front cover 10.1039/c1md90025k AuthorAnonymous 2011 2 8 677 678 Abstract HTML PDF other

MedChemComm 2040-2503 Royal Society of Chemistry Contents list 10.1039/c1md90028e AuthorAnonymous 2011 2 8 679 688 Abstract HTML PDF other

MedChemComm 2040-2503 Royal Society of Chemistry Progress on lamellarins 10.1039/c1md00003a Pla Daniel Albericio Fernando Álvarez Mercedes 2011 2 8 689 697 Abstract HTML PDF review-article

MedChemComm 2040-2503 Royal Society of Chemistry Nitro-based inhibitors against thermolysin 10.1039/c1md00088h Tian Guan Rong Wang Si-Hong Wang Shou-Feng Meng Ling-Qiang Li Hui Zeng Zong-Hao Jin 2011 2 8 698 700 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry HIV-1 protease inhibitors with a tertiary alcohol containing transition-state mimic and various P2 and P1′ substituents 10.1039/c1md00077b Öhrngren Per Wu Xiongyu Persson Magnus Ekegren Jenny K. Wallberg Hans Vrang Lotta Rosenquist Åsa Samuelsson Bertil Unge Torsten Larhed Mats 2011 2 8 701 709 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry Determination of structural requirements of influenza neuraminidase type A inhibitors and binding interaction analysis with the active site of A/H1N1 by 3D-QSAR CoMFA and CoMSIA modeling 10.1039/c1md00050k Murumkar Prashant R. Le Ly Truong Thanh N. Yadav Mange Ram 2011 2 8 710 719 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry Metal preference of Zn(ii) and Co(ii) for the dinuclear metal binding site of IMP-1 metallo-β-lactamase and spectroscopic properties of Co(ii)-substituted IMP-1 with mercaptoacetic acid 10.1039/c1md00062d Yamaguchi Yoshihiro Imamura Kayo Sasao Ako Murakami Emi Arakawa Yoshichika Kurosaki Hiromasa 2011 2 8 720 725 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry Beta-adrenergic receptor signaling by the isomers of isoproterenol and like drugs in retinal endothelial cells and Müller cells 10.1039/c0md00227e Pagadala Jayaprakash Williams-Guy Kimberly Nooh Mohammed M. Steinle Jena J. Miller Duane D. 2011 2 8 726 730 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry Effect of the isosteric replacement of the phenyl motif with furyl (or thienyl) of 4-phenyl-<i>N</i>-arylsulfonylimidazolones as broad and potent anticancer agents 10.1039/c0md00219d Sharma Vinay K. Hung Dang The Lee Ki-Cheul Thanigaimalai P. Kang Jong Seong Kim Hwan-Mook Jung Sang-Hun 2011 2 8 731 734 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry New analyses of MIC₉₀ data to aid antibacterial drug discovery 10.1039/c1md00095k Brown Matthew F. Gupta Rishi R. Kuhn Max Flanagan Mark E. Mitton-Fry Mark 2011 2 8 735 742 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry Synthesis and biological activity evaluation of <i>N</i>-protected isatin derivatives as inhibitors of ICAM-1 expression on human endothelial cells 10.1039/c0md00262c Malhotra Shashwat Balwani Sakshi Dhawan Ashish Singh Brajendra K. Kumar Sarvesh Thimmulappa Rajesh Biswal Shyam Olsen Carl E. Eycken Erik Van der Prasad Ashok K. Ghosh Balaram Parmar Virinder S. 2011 2 8 743 751 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry Structure–activity relationship of conformationally constrained peptidomimetics for antiproliferative activity in HER2-overexpressing breast cancer cell lines 10.1039/c1md00126d Banappagari Sashikanth Ronald Sharon Satyanarayanajois Seetharama D. 2011 2 8 752 759 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry Potent and selective inhibitors of human peptidylglycine α-amidating monooxygenase 10.1039/c1md00079a Cao Feihua Gamble Allan B. Kim Hye-Kyung Onagi Hideki Gresser Mary J. Kerr Jamie Easton Christopher J. 2011 2 8 760 763 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry Blockage of collagen binding to integrin α2β1: structure–activity relationship of protein–protein interaction inhibitors 10.1039/c1md00089f Koivunen Jarkko T. Nissinen Liisa Juhakoski Auni Pihlavisto Marjo Marjamäki Anne Huuskonen Juhani Pentikäinen Olli T. 2011 2 8 764 770 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry Overcoming retinoic acid receptor-α based testicular toxicity in the optimisation of glucokinase activators 10.1039/c1md00090j Waring Michael J. Brogan Iain J. Coghlan Matthew Johnstone Craig Jones Huw B. Leighton Brendan McKerrecher Darren Pike Kurt G. Robb Graeme R. 2011 2 8 771 774 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry Matrix-based multiparameter optimisation of glucokinase activators: the discovery of <b>AZD1092</b> 10.1039/c1md00092f Waring Michael J. Johnstone Craig McKerrecher Darren Pike Kurt G. Robb Graeme 2011 2 8 775 779 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry Carbazole–pyrrolo[2,1-<i>c</i>][1,4]benzodiazepine conjugates: design, synthesis, and biological evaluation 10.1039/c1md00072a Kamal Ahmed Shetti Rajesh V. C. R. N. C. Ramaiah M. Janaki Swapna P. Reddy K. Srinivasa Mallareddy A. Rao M. P. Narasimha Chourasia Mukesh Sastry G. Narahari Juvekar Aarti Zingde Surekha Sarma Pranjal Pushpavalli S. N. C. V. L. Pal-Bhadra Manika 2011 2 8 780 788 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry Novel <i>N</i>-sulfonamide <i>trans</i>-platinum complexes: synthesis, reactivity and <i>in vitro</i> evaluation 10.1039/c1md00070e Alemán José Solar Virginia del Alvarez-Valdés Amparo Ríos-Luci Carla Padrón José M. Navarro-Ranninger Carmen 2011 2 8 789 793 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry Structure-based design, synthesis, and profiling of a β-tryptase inhibitor with a spiro-piperidineamide scaffold, benzylamine P1 group, and a substituted indole P4 group 10.1039/c1md00104c Liang Guyan Choi-Sledeski Yong Mi Poli Gregory B. Chen Xin Minnich Anne Wang Qingping Tsay Joseph Sides Keith Vaz Roy J. 2011 2 8 794 799 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry Peptidomimetic nitriles as selective inhibitors for the malarial cysteine protease falcipain-2 10.1039/c1md00115a Ehmke Veronika Kilchmann Falco Heindl Cornelia Cui Kunqiang Huang Jin Schirmeister Tanja Diederich François 2011 2 8 800 804 Abstract HTML PDF research-article

MedChemComm 2040-2503 Royal Society of Chemistry MedChemWatch Issue 13 and Back matter 10.1039/c1md90026a AuthorAnonymous 2011 2 8 805 806 Abstract HTML PDF other

MedChemComm 2040-2503 Royal Society of Chemistry Back cover 10.1039/c1md90027g AuthorAnonymous 2011 2 8 807 808 Abstract HTML PDF other