MedChemComm
2040-2503
Royal Society of Chemistry
Front cover
10.1039/C8MD90053A
AuthorAnonymous
2018
9
12
1975
1976
Abstract
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MedChemComm
2040-2503
Royal Society of Chemistry
Contents list
10.1039/C8MD90054J
AuthorAnonymous
2018
9
12
1977
1982
Abstract
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MedChemComm
2040-2503
Royal Society of Chemistry
The transition to magic bullets – transition state analogue drug design
10.1039/c8md00372f
Evans
Gary B.
Schramm
Vern L.
Tyler
Peter C.
2018
9
12
1983
1993
Abstract
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review-article
MedChemComm
2040-2503
Royal Society of Chemistry
Flush with a flash: natural three-component antimicrobial combinations based on <i>S</i>-nitrosothiols, controlled superoxide formation and “domino” reactions leading to peroxynitrite
10.1039/c8md00414e
Alhasan
Rama
Kharma
Ammar
Nasim
Muhammad Jawad
Abdin
Ahmad Yaman
Bonetti
Justine
Giummelly
Philippe
Ejike
Chukwunonso E. C. C.
Leroy
Pierre
Gaucher
Caroline
Jacob
Claus
2018
9
12
1994
1999
Abstract
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research-article
MedChemComm
2040-2503
Royal Society of Chemistry
Probing the <i>hras</i>-1<sup>Y</sup> i-motif with small molecules
10.1039/c8md00311d
Journey
Sara N.
Alden
Stephanie L.
Hewitt
Will M.
Peach
Megan L.
Nicklaus
Marc C.
Jr
John S. Schneekloth
2018
9
12
2000
2007
Abstract
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research-article
MedChemComm
2040-2503
Royal Society of Chemistry
Structure–activity relationship of the cinnamamide family of antibiotic potentiators for methicillin-resistant <i>Staphylococcus aureus</i> (MRSA)
10.1039/c8md00479j
Speri
Enrico
Fishovitz
Jennifer
Mobashery
Shahriar
2018
9
12
2008
2016
Abstract
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research-article
MedChemComm
2040-2503
Royal Society of Chemistry
Novel <i>O</i>-methyl goniofufurone and 7-<i>epi</i>-goniofufurone derivatives: synthesis, <i>in vitro</i> cytotoxicity and SAR analysis
10.1039/c8md00431e
Francuz
Jovana
Popsavin
Mirjana
Djokić
Sanja
Kojić
Vesna
Srdić-Rajić
Tatjana
Rodić
Marko V.
Jakimov
Dimitar
Popsavin
Velimir
2018
9
12
2017
2027
Abstract
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research-article
MedChemComm
2040-2503
Royal Society of Chemistry
Discovery of 3-hydroxy-3-pyrrolin-2-one-based mPGES-1 inhibitors using a multi-step virtual screening protocol
10.1039/c8md00497h
Lauro
Gianluigi
Cantone
Vincenza
Potenza
Marianna
Fischer
Katrin
Koeberle
Andreas
Werz
Oliver
Riccio
Raffaele
Bifulco
Giuseppe
2018
9
12
2028
2036
Abstract
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research-article
MedChemComm
2040-2503
Royal Society of Chemistry
Screening of the Pathogen Box reveals new starting points for anti-trypanosomal drug discovery
10.1039/c8md00319j
Veale
Clinton G. L.
Hoppe
Heinrich C.
2018
9
12
2037
2044
Abstract
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research-article
MedChemComm
2040-2503
Royal Society of Chemistry
Exploring the effectiveness of novel benzimidazoles as CB2 ligands: synthesis, biological evaluation, molecular docking studies and ADMET prediction
10.1039/c8md00461g
Tonelli
Michele
Cichero
Elena
Mahmoud
Alì Mokhtar
Rabbito
Alessandro
Tasso
Bruno
Fossa
Paola
Ligresti
Alessia
2018
9
12
2045
2054
Abstract
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research-article
MedChemComm
2040-2503
Royal Society of Chemistry
Development of selective, fluorescent cannabinoid type 2 receptor ligands based on a 1,8-naphthyridin-2-(1<i>H</i>)-one-3-carboxamide scaffold
10.1039/c8md00448j
Cooper
Anna G.
Oyagawa
Caitlin R. M.
Manning
Jamie J.
Singh
Sameek
Hook
Sarah
Grimsey
Natasha L.
Glass
Michelle
Tyndall
Joel D. A.
Vernall
Andrea J.
2018
9
12
2055
2067
Abstract
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research-article
MedChemComm
2040-2503
Royal Society of Chemistry
A β-glucuronidase-responsive albumin-binding prodrug programmed for the double release of monomethyl auristatin E
10.1039/c8md00466h
Renoux
Brigitte
Fangous
Laure
Hötten
Camille
Péraudeau
Elodie
Eddhif
Balkis
Poinot
Pauline
Clarhaut
Jonathan
Papot
Sébastien
2018
9
12
2068
2071
Abstract
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research-article
MedChemComm
2040-2503
Royal Society of Chemistry
Synthesis of d-(+)-camphor-based <i>N</i>-acylhydrazones and their antiviral activity
10.1039/c8md00442k
Kovaleva
Kseniya S.
Zubkov
Fedor I.
Bormotov
Nikolay I.
Novikov
Roman A.
Dorovatovskii
Pavel V.
Khrustalev
Victor N.
Gatilov
Yuriy V.
Zarubaev
Vladimir V.
Yarovaya
Olga I.
Shishkina
Larisa N.
Salakhutdinov
Nariman F.
2018
9
12
2072
2082
Abstract
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research-article
MedChemComm
2040-2503
Royal Society of Chemistry
Discovery of a 3,4,5-trisubstituted-1,2,4-triazole agonist with high affinity and selectivity at the somatostatin subtype-4 (sst<sub>4</sub>) receptor
10.1039/c8md00388b
Daryaei
Iman
Sandoval
Karin
Witt
Ken
Kontoyianni
Maria
Crider
A. Michael
2018
9
12
2083
2090
Abstract
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research-article
MedChemComm
2040-2503
Royal Society of Chemistry
Synthesis and potential antineoplastic activity of dehydroabietylamine imidazole derivatives
10.1039/c8md00487k
Zhao
Fengyi
Lu
Wen
Su
Fan
Xu
Li
Jiang
Dong
Sun
Xu
Shi
Jiuzhou
Zhou
Mengyi
Lin
Feng
Cao
Fuliang
2018
9
12
2091
2099
Abstract
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research-article
MedChemComm
2040-2503
Royal Society of Chemistry
Novel benzoyl thioureido benzene sulfonamides as highly potent and selective inhibitors of carbonic anhydrase IX: optimization and bioactive studies
10.1039/c8md00392k
Liu
Li
Wang
Wanqi
Huang
Jin
Zhao
Zhenjiang
Li
Honglin
Xu
Yufang
2018
9
12
2100
2105
Abstract
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research-article
MedChemComm
2040-2503
Royal Society of Chemistry
Design, synthesis, and biological activity of novel ammonium salts containing sterically hindered phenolic fragment and phosphoryl group
10.1039/c8md00481a
Starodubtseva
Ramilya R.
Gibadullina
Elmira M.
Pazilova
Nurbala B.
Sapunova
Anastasiia S.
Voloshina
Alexandra D.
Sudakov
Igor A.
Vyshtakalyuk
Alexandra B.
Pudovik
Michael A.
Burilov
Alexander R.
Bukharov
Sergey V.
2018
9
12
2106
2120
Abstract
HTMLPDF
research-article
MedChemComm
2040-2503
Royal Society of Chemistry
Correction: Synthesis and anticonvulsant activity of phenoxyacetyl derivatives of amines, including aminoalkanols and amino acids
10.1039/c8md90052c
Pańczyk
Katarzyna
Żelaszczyk
Dorota
Koczurkiewicz
Paulina
Słoczyńska
Karolina
Pękala
Elżbieta
Żesławska
Ewa
Nitek
Wojciech
Żmudzki
Paweł
Marona
Henryk
Waszkielewicz
Anna
2018
9
12
2121
2121
Abstract
HTML
PDF
research-article
MedChemComm
2040-2503
Royal Society of Chemistry
Back cover
10.1039/C8MD90055H
AuthorAnonymous
2018
9
12
2123
2124
Abstract
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